Apicomplexan parasites: molecular approaches toward targeted drug development
Gespeichert in:
Weitere beteiligte Personen: | |
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Format: | Buch |
Sprache: | Englisch |
Veröffentlicht: |
Weinheim
Wiley-Blackwell
2011
|
Schriftenreihe: | Drug discovery in infectious diseases
2 |
Schlagwörter: | |
Links: | http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=024989684&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
Umfang: | XXI, 528 S. Ill., graph. Darst. |
ISBN: | 9783527327317 3527327312 |
Internformat
MARC
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---|---|---|---|
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245 | 1 | 0 | |a Apicomplexan parasites |b molecular approaches toward targeted drug development |c ed. by Katja Becker |
264 | 1 | |a Weinheim |b Wiley-Blackwell |c 2011 | |
300 | |a XXI, 528 S. |b Ill., graph. Darst. | ||
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650 | 0 | 7 | |a Arzneimittelentwicklung |0 (DE-588)4143176-5 |2 gnd |9 rswk-swf |
653 | |a Protozoan vaccines / Development | ||
653 | |a Apicomplexa | ||
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Datensatz im Suchindex
_version_ | 1819322825182281728 |
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adam_text | IMAGE 1
VII
CONTENTS
FOREWORD V PREFACE XI
LIST OF CONTRIBUTORS XIII
PART ONE SCREENING, BIOINFORMATICS, CHEMOINFORMATICS, AND DRUG DESIGN 1
1 DRUG DISCOVERY APPROACHES TOWARD ANTI-PARASITIC AGENTS 3 ANDREAS
ROHWER, RICHARDJ. MARHOEFER, CONOR R. CAFFREY, AND PAUL M. SEHER
2 NEW BIOINFORMATIC STRATEGIES AGAINST APICOMPLEXAN PARASITES 21 THOMAS
DANDEKAR AND KE XIAO
3 SORTING POTENTIAL THERAPEUTIC TARGETS IN APICOMPLEXA 35 JAN A. HISS
AND CISBERT SCHNEIDER
4 ALTERNATIVES TO DRUG DEVELOPMENT IN THE APICOMPLEXA 53 THEO P.M.
SCHETTERS
PART TWO METABOLIC PATHWAYS AND PROCESSES ADDRESSED BY CURRENT
DRUG-DISCOVERY APPROACHES 75
5 ENERGY METABOLISM AS AN ANTIMALARIAL DRUG TARGET 77 ESTHERJORTZIK AND
KATJA BECKER
6 POLYAMINES IN APICOMPLEXAN PARASITES 97 INGRID B. MUELLER, ROBIN DAS
GUPTA, KAI LUEERSEN, CARSTEN WRENGER, AND ROLFD. WALTER
BIBLIOGRAFISCHE INFORMATIONEN HTTP://D-NB.INFO/1006150196
DIGITALISIERT DURCH
IMAGE 2
VIII I CONTENTS
7 THE REDUCING MILIEU OF PARASITIZED CELLS AS A TARGET OF ANTIMALARIAL
AGENTS: METHYLENE BLUE AS AN ETHICAL DRUG 215 PETER MEISSNER, HEIKE
ADLER, DENIS KASOZI, KARIN FRITZ-WOLF AND R. HEINER SCHIRMER
8 LIPIDS AS DRUG TARGETS FOR MALARIA THERAPY 137
HENRIJ. VIAL, DIANA PENARETE, SHARON WEIN, SERGIO CALDARELLI, LAURENT
FRAISSE, AND SUZANNE PEYROTTES
9 TARGETING APICOPLAST PATHWAYS IN PLASMODIUM 163 SNOBER S. MIR, SUBIR
BISWAS, AND SAMAN HABIB
10 LIPOIC ACID ACQUISITION AND CLUTATHIONE BIOSYNTHESIS IN APICOMPLEXAN
PARASITES 187 JANET STORM, EVA-MARIA PATZEWITZ, AND SYLKE MUELLER
11 ANTIMALARIAL DRUGS AND MOLECULES INHIBITING HEMOZOIN FORMATION 205
UDAY BANDYOPADHYAY AND SUMANTA DEY
12 EXPLOITING THE VITAMIN METABOLISM OF APICOMPLEXA AS DRUG TARGETS 235
CARSTEN WRENGER AND INGRID B. MUELLER
13 VITAMIN BIOSYNTHETIC PATHWAYS, THE PLP SYNTHASE COMPLEX, AND THE
POTENTIAL FOR TARGETING PROTEIN-PROTEIN INTERACTION 251 IVO TEWS AND
IRMGARD SINNING
14 TARGETING PROKARYOTIC ENZYMES IN THE EUKARYOTIC PATHOGEN
CRYPTOSPORIDIUM 271 SURESH KUMAR CORLA, COREY JOHNSON, JIHAN KHAN, XIN
SUN, LISA SHARLING, BORIS STRIEPEN, AND LIZBETH HEDSTROM
PART THREE DRUG TARGETS IN APICOMPLEXAN PARASITES 287
15 NOVEL APICOMPLEXAN PHOSPHATASES AND IMMUNOPHILINS AS DOMAIN-SPECIFIC
DRUG TARGETS 289 SAILEN BARIK
16 DEHYDROGENASES AND ENZYMES OF THE MITOCHONDRIAL ELECTRON TRANSPORT
CHAIN AS ANTI-APICOMPLEXAN DRUG TARGETS 307 KATHLEEN ZOCHER, STEFAN
RAHLFS, AND KATJA BECKER
17 CALCIUM-DEPENDENT PROTEIN KINASES AS DRUG TARGETS IN APICOMPLEXAN
PARASITES 319 DOMINIK KUGELSTADT, BIANCA DERRER, AND BARBARA KAPPES
IMAGE 3
CONTENTS IX
18 PROTEIN ACYLATION: NEW POTENTIAL TARGETS FOR INTERVENTION
AGAINST THE APICOMPLEXA 335 JOANA M. SANTOS, CHRISTIAN HEDBERG, AND
DOMINIQUE SOLDATI-FAVRE
19 DRUGS AND DRUG TARGETS IN NEOSPORA CANINUM AND RELATED APICOMPLEXANS
359 JOACHIM MUELLER, NORBERT MUELLER, AND ANDREW HEMPHILL
PART FOUR COMPOUNDS 373
20 SUBVERSIVE SUBSTRATES OF CLUTATHIONE REDUCTASES FROM PLASMODIUM
FALCIPARUM- NFECTED RED BLOOD CELLS AS ANTIMALARIAL AGENTS 375 ELISABETH
DAVIOUD-CHARVET AND DON ANTOINE LANFRANCHI
21 FERROQUINE: A CONCEALED WEAPON 397 CHRISTOPHE BIOT, BRUNO PRADINES,
AND DANIEL DIVE
22 CURRENT ASPECTS OF ENDOPEROXIDES IN ANTIPARASITIC CHEMOTHERAPY 413
DENIS MATOVU KASOZI, STEFAN RAHLFI, AND KATJA BECKER
23 PLASMODIUM HSP90 AS AN ANTIMALARIAL TARGET 431 C. SRIDHAR PRASAD,
NICHOLAS D.P. COSFORD, AND SAILEN BARIK
24 DRUG DISCOVERY AGAINST BABESIA AND TOXOPLASMA 453 MOHAMAD ALAA
TERKAWI AND IKUO IGARASHI
25 SEARCH FOR DRUGS AND DRUG TARGETS AGAINST BABESIA BOVIS, BABESIA
BIGEMINA, BABESIA CABALLI, AND BABESIA [THEILERIA) EQUI 469 SABINE
BORK-MIMM
26 ORLISTAT: A REPOSITIONING OPPORTUNITY AS A GROWTH INHIBITOR OF
APICOMPLEXAN PARASITES? 481 CHRISTIAN MICULKA, HON Q. TRAN, THORSTEN
MEYER, ANJA R. HECKEROTH, STEFAN BAUMEISTER, FRANK SEEBER, AND PAUL M.
SELZER
27 RECENT DRUG DISCOVERY AGAINST CRYPTOSPORIDIUM 493 JEAN-FRANGOIS
ROSSIGNOL,J. EDWARD SEMPLE, ANDREW V. STACHULSKI, AND CILLES GARGALA
INDEX 513
|
any_adam_object | 1 |
author2 | Becker, Katja 1965- |
author2_role | edt |
author2_variant | k b kb |
author_GND | (DE-588)120316390 |
author_facet | Becker, Katja 1965- |
building | Verbundindex |
bvnumber | BV040132559 |
classification_rvk | XX 3000 |
ctrlnum | (OCoLC)724747271 (DE-599)BSZ336165536 |
dewey-full | 615.19 |
dewey-hundreds | 600 - Technology (Applied sciences) |
dewey-ones | 615 - Pharmacology and therapeutics |
dewey-raw | 615.19 |
dewey-search | 615.19 |
dewey-sort | 3615.19 |
dewey-tens | 610 - Medicine and health |
discipline | Medizin |
format | Book |
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genre | (DE-588)4143413-4 Aufsatzsammlung gnd-content |
genre_facet | Aufsatzsammlung |
id | DE-604.BV040132559 |
illustrated | Illustrated |
indexdate | 2024-12-20T16:08:51Z |
institution | BVB |
isbn | 9783527327317 3527327312 |
language | English |
oai_aleph_id | oai:aleph.bib-bvb.de:BVB01-024989684 |
oclc_num | 724747271 |
open_access_boolean | |
owner | DE-11 |
owner_facet | DE-11 |
physical | XXI, 528 S. Ill., graph. Darst. |
publishDate | 2011 |
publishDateSearch | 2011 |
publishDateSort | 2011 |
publisher | Wiley-Blackwell |
record_format | marc |
series | Drug discovery in infectious diseases |
series2 | Drug discovery in infectious diseases |
spellingShingle | Apicomplexan parasites molecular approaches toward targeted drug development Drug discovery in infectious diseases Parasitäre Krankheit (DE-588)4044638-4 gnd Sporentierchen (DE-588)4319742-5 gnd Arzneimittelentwicklung (DE-588)4143176-5 gnd |
subject_GND | (DE-588)4044638-4 (DE-588)4319742-5 (DE-588)4143176-5 (DE-588)4143413-4 |
title | Apicomplexan parasites molecular approaches toward targeted drug development |
title_auth | Apicomplexan parasites molecular approaches toward targeted drug development |
title_exact_search | Apicomplexan parasites molecular approaches toward targeted drug development |
title_full | Apicomplexan parasites molecular approaches toward targeted drug development ed. by Katja Becker |
title_fullStr | Apicomplexan parasites molecular approaches toward targeted drug development ed. by Katja Becker |
title_full_unstemmed | Apicomplexan parasites molecular approaches toward targeted drug development ed. by Katja Becker |
title_short | Apicomplexan parasites |
title_sort | apicomplexan parasites molecular approaches toward targeted drug development |
title_sub | molecular approaches toward targeted drug development |
topic | Parasitäre Krankheit (DE-588)4044638-4 gnd Sporentierchen (DE-588)4319742-5 gnd Arzneimittelentwicklung (DE-588)4143176-5 gnd |
topic_facet | Parasitäre Krankheit Sporentierchen Arzneimittelentwicklung Aufsatzsammlung |
url | http://bvbr.bib-bvb.de:8991/F?func=service&doc_library=BVB01&local_base=BVB01&doc_number=024989684&sequence=000001&line_number=0001&func_code=DB_RECORDS&service_type=MEDIA |
volume_link | (DE-604)BV040160480 |
work_keys_str_mv | AT beckerkatja apicomplexanparasitesmolecularapproachestowardtargeteddrugdevelopment |